ISENTRESS (Raltegravir)

ISENTRESS (Raltegravir) is an antiretroviral medication used in the treatment of HIV-1 infection. It belongs to a class of drugs known as integrase inhibitors, which work by blocking the integration of viral DNA into the host cell's DNA, thereby preventing the replication of the virus.

This medication is typically prescribed as part of a comprehensive HIV treatment regimen, often in combination with other antiretroviral agents to enhance efficacy and reduce viral load. ISENTRESS is effective in both treatment-naive patients and those who have previously been treated for HIV.

Some key highlights of ISENTRESS include:

• Efficacy: Clinical studies have shown that ISENTRESS effectively reduces viral load, helping patients achieve and maintain undetectable levels of HIV in their blood.


• Safety: ISENTRESS is generally well-tolerated, with a favorable safety profile. Common side effects may include headache, insomnia, and gastrointestinal issues.


• Convenience: Available in both tablet and chewable forms, ISENTRESS offers flexible dosing options, making it easier for patients to adhere to their treatment plans.


• Resistance Profile: Raltegravir has a low barrier to resistance, meaning that it remains effective even in patients with some resistance mutations.


• Pregnancy Category: It is categorized as pregnancy category B, indicating that it is considered safe for use during pregnancy based on available studies.

Patients considering ISENTRESS should consult with their healthcare provider to discuss potential benefits, risks, and how it fits into their overall treatment strategy for managing HIV. Regular monitoring and follow-up are essential to ensure optimal therapeutic outcomes.

• Raltegravir


• Microcrystalline cellulose


• Pregelatinized starch


• Croscarmellose sodium


• Magnesium stearate


• Silicon dioxide


• Coating: Hypromellose


• Macrogol


• Titanium dioxide


• Iron oxide

ISENTRESS (Raltegravir) is an antiretroviral medication used to treat HIV infection. To use this medication effectively, follow these guidelines:

1. Consult Your Healthcare Provider: Before starting ISENTRESS, discuss your medical history and any other medications you are taking with your healthcare provider to ensure it is a suitable option for you.


2. Dosage Instructions: Take ISENTRESS exactly as prescribed by your doctor. The typical dosage for adults is 400 mg taken twice daily.


3. Administration: You can take ISENTRESS with or without food. Swallow the tablets whole with a glass of water. Do not chew or crush the tablets.


4. Missed Dose: If you miss a dose, take it as soon as you remember. If it's almost time for your next dose, skip the missed dose. Never take two doses at the same time to make up for a missed one.


5. Side Effects: Be aware of potential side effects, which may include nausea, headache, or insomnia. If you experience severe side effects, such as allergic reactions or muscle pain, contact your healthcare provider immediately.


6. Regular Monitoring: Attend regular follow-up appointments with your healthcare provider to monitor your response to the medication and any potential side effects.


7. Adherence: It is crucial to adhere to the prescribed regimen to maintain the effectiveness of the treatment and prevent the development of drug resistance.


8. Storage: Store ISENTRESS at room temperature, away from moisture and heat. Keep it out of reach of children.

By following these instructions and maintaining open communication with your healthcare provider, you can effectively manage your HIV treatment with ISENTRESS.